Detalhe da pesquisa
1.
N-substituted 2-isonicotinoylhydrazinecarboxamides--new antimycobacterial active molecules.
Molecules
; 19(4): 3851-68, 2014 Mar 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-24686575
2.
Diethyl 2-(phenylcarbamoyl)phenyl phosphorothioates: synthesis, antimycobacterial activity and cholinesterase inhibition.
Molecules
; 19(6): 7152-68, 2014 May 30.
Artigo
em Inglês
| MEDLINE | ID: mdl-24886941
3.
Preparation, in vitro evaluation and molecular modelling of pyridinium-quinolinium/isoquinolinium non-symmetrical bisquaternary cholinesterase inhibitors.
Bioorg Med Chem Lett
; 23(24): 6663-6, 2013 Dec 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-24220173
4.
Preparation, in vitro screening and molecular modelling of symmetrical bis-quinolinium cholinesterase inhibitors--implications for early myasthenia gravis treatment.
Bioorg Med Chem Lett
; 21(8): 2505-9, 2011 Apr 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-21397501
5.
Preparation, in vitro screening and molecular modelling of symmetrical 4-tert-butylpyridinium cholinesterase inhibitors--analogues of SAD-128.
Bioorg Med Chem Lett
; 21(1): 150-4, 2011 Jan 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21144749
6.
Mono-oxime bisquaternary acetylcholinesterase reactivators with prop-1,3-diyl linkage-Preparation, in vitro screening and molecular docking.
Bioorg Med Chem
; 19(2): 754-62, 2011 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-21215642
7.
The preparation, in vitro screening and molecular docking of symmetrical bisquaternary cholinesterase inhibitors containing a but-(2E)-en-1,4-diyl connecting linkage.
J Enzyme Inhib Med Chem
; 26(2): 245-53, 2011 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-21406034
8.
Preparation and in vitro screening of symmetrical bispyridinium cholinesterase inhibitors bearing different connecting linkage-initial study for Myasthenia gravis implications.
Bioorg Med Chem Lett
; 20(5): 1763-6, 2010 Mar 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20138518
9.
Preparation and in vitro screening of symmetrical bis-isoquinolinium cholinesterase inhibitors bearing various connecting linkage--implications for early Myasthenia gravis treatment.
Eur J Med Chem
; 46(2): 811-8, 2011 Feb.
Artigo
em Inglês
| MEDLINE | ID: mdl-21236521